99% Tianeptine sodium mchere CAS 30123-17-2
Kufotokozera
ITEM | ZOYENERA | ZOtsatira |
Maonekedwe | Ufa woyera mpaka wachikasu | White crystalline ufa |
Kusungunuka | Momasuka sungunuka M'madzi ndi methanol ndi dichloromethane | Zimagwirizana |
Chizindikiritso | Ndi IR, Kufananiza ndi mulingo wogwirira ntchito | Zimagwirizana |
(2) Amapereka kuyankha kwa sodium | Zimagwirizana | |
Zonyansa A | ≤0.1% | Sizinazindikirike |
Zosakaniza zogwirizana | Chidetso chilichonse cha Max Chilichonse≤0.1% | 0.060% |
Zonyansa zonse≤0.4% | 0.36% | |
Zosungunulira Zotsalira (GC) | Acetidin ≤ 0.5% | ND |
Dichloromethane ≤ 0.06% | ND | |
Methanol ≤ 0.3% | ND | |
Acetone ≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.022% | |
Ethanol ≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Madzi | ≤ 5.0% | 3.8% |
Kuyesa (HPLC) | 99.0% -101.0% (Pa anhydrousbasis) | 99.70% |
Kugwiritsa ntchito
Tianeptine sodiummcherendi tricyclic antidepressant.Kachitidwe kake ka antidepressant ndi kosiyana ndi kachitidwe ka tricyclic antidepressants.Ikhoza kuonjezera kubwereza kwa 5-HT mu synaptic cleft.Zotsatira za HT neuronal conduction.Palibe kuyanjana kwa choline kapena adrenergic receptors.Mphamvu ya antidepressant ndi yofanana ndi ya tricyclics, koma kulekerera ndikwabwino kuposa tricyclics.Pochiza kukhumudwa pang'ono, pang'onopang'ono kapena koopsa, kupsinjika kwa neuroogenic ndi kuchitapo kanthu, nkhawa ndi kupsinjika ndi thupi, makamaka kusapeza bwino kwa m'mimba, komanso nkhawa ndi kupsinjika kwa odwala omwe amamwa mowa panthawi yosiya.